1. Signaling Pathways
  2. Epigenetics
  3. Histone Demethylase
  4. Histone Demethylase Inhibitors

Histone Demethylase Inhibitors

KDM1/LSD1

KDM2

KDM3

KDM4

KDM5

KDM6

KDM7

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Sorry. There is currently no product that acts on isoform together.

Please try each isoform separately.

Histone Demethylase Inhibitors & Antagonists
Product Name KDM1/LSD1 KDM2 KDM3 KDM4 KDM5 KDM6 KDM7 Purity
GSK-J4          
KDM6
  99.64%
CPI-455        
KDM5
    98.95%
IOX1  
KDM2
KDM3
KDM4
 
KDM6
  99.89%
GSK2879552
KDM1/LSD1
            99.90%
JIB-04      
KDM4
KDM5
KDM6
  98.29%
Iadademstat dihydrochloride
KDM1/LSD1
            99.98%
GSK-J1          
KDM6
  99.94%
KDM5-C70        
KDM5
   
QC6352      
KDM4A, IC50: 104 nM
KDM4B, IC50: 56 nM
KDM4C, IC50: 35 nM
KDM4D, IC50: 104 nM
KDM5B, IC50: 750 nM
    99.13%
GSK-J4 hydrochloride          
KDM6
  99.01%
GSK-LSD1 dihydrochloride
KDM1/LSD1
            ≥98.0%
SP2509
KDM1/LSD1
            99.90%
Tranylcypromine hemisulfate
KDM1/LSD1
            99.94%
Seclidemstat
KDM1/LSD1
            99.77%
GSK467        
KDM5, Ki: 10 nM
KDM5, IC50: 26 nM
    99.55%
Daminozide  
KDM2
          99.79%
AS8351        
KDM5
    99.88%
KDOAM-25 citrate        
KDM5
    98.56%
ML324      
KDM4
      98.46%
Pulrodemstat benzenesulfonate
KDM1/LSD1
            99.64%
NCGC00244536      
KDM4
      99.70%
KDM5A-IN-1        
KDM5
    99.64%
Bomedemstat ditosylate
KDM1/LSD1
            99.14%
PFI-90    
KDM3
        99.86%
Bomedemstat hydrochloride
KDM1/LSD1
            99.94%
TK-129        
KDM5, IC50: 44 nM
    ≥98.0%
Iadademstat
LSD1
            99.82%
KDM2A/7A-IN-1  
KDM2
          99.94%
Bomedemstat dihydrochloride
KDM1/LSD1
            99.55%
KDM2/7-IN-1  
KDM2
 
KDM4
   
KDM7
99.00%
KDM5-IN-1        
KDM5
    99.52%
TAK-418
KDM1/LSD1
            99.81%
KDM4D-IN-1      
KDM4
      98.82%
KDM4C-IN-1      
KDM4
      98.13%
PBIT        
KDM5
    99.46%
Seclidemstat mesylate
KDM1/LSD1
            99.80%
S2101
KDM1/LSD1
            99.70%
NSC636819      
KDM4
      98.90%
DDP-38003 dihydrochloride
KDM1/LSD1
            98.22%
GSK 690 Hydrochloride
KDM1/LSD1
            98.58%
KDM4-IN-3      
KDM4
      99.36%
T-3775440 hydrochloride
KDM1/LSD1
            99.13%
JQKD82 trihydrochloride        
KDM5
    99.94%
KDM2B-IN-4  
KDM2
          99.61%
YUKA1        
KDM5
    99.56%
INCB059872 dihydrochloride
KDM1/LSD1
            99.18%
LSD1/HDAC6-IN-2
LSD1, IC50: 5 nM
            99.66%
DDP-38003 trihydrochloride
KDM1/LSD1
           
INCB059872
KDM1/LSD1
            98.06%
HDAC6-IN-3
KDM1/LSD1
            ≥98.0%
LSD1-IN-30
LSD1, IC50: 0.291 μM
            99.03%
CBB1007 trihydrochloride
KDM1/LSD1
           
Pulrodemstat
KDM1/LSD1
           
Bomedemstat
KDM1/LSD1
            98.23%
KDM4-IN-2      
KDM4
      98.29%
Arborinine
LSD1
            99.87%
NCGC00247743      
KDM4
      98.61%
CBB1007 hydrochloride
KDM1/LSD1
            ≥98.0%
GSK-J1 lithium salt          
KDM6
  98.33%
LSD1-IN-5
KDM1/LSD1
           
LSD1-IN-6
KDM1/LSD1
           
Pulrodemstat Methylbenzenesulfonate
KDM1/LSD1
           
CPI-455 hydrochloride        
KDM5
   
LSD1/HDAC6-IN-1
KDM1/LSD1
           
LSD1-IN-13 hydrochloride
KDM1/LSD1
           
MC2652
KDM1/LSD1
           
KDM4-IN-4      
KDM4A-Tudor domain, Ki: 80 μM
     
LSD1-IN-31
LSD1
           
LSD1-IN-34
LSD1, IC50: 4.51 nM
           
HSP90/LSD1-IN-1
LSD1
           
LSD1-UM-109
LSD1, IC50: 3.1 nM
           
LSD1-IN-38
LSD1, IC50: 1.2 nM
           
S1427
KDM1/LSD1
           
LSD1-IN-23
KDM1/LSD1, IC50: 0.58 μM
           
LSD1/2-IN-4
KDM1/LSD1
           
NCL1
LSD1, IC50: 2.5 ± 0.5 μM
           
cis-4-Br-2,5-F2-PCPA
KDM1/LSD1
           
KDM1/CDK1-IN-1
KDM1/LSD1
           
LSD1/HDAC-IN-2
KDM1/LSD1, IC50: 39.0 nM
           
LSD1-IN-26
LSD1, IC50: 25.3 ± 1.4 nM
           
LSD1-IN-21
LSD1, IC50: 0.956 μM
           
KDM5-C49        
KDM5
   
LSD1-IN-35
LSD1
           
LSD1-IN-18
KDM1/LSD1
           
LSD1-IN-25
LSD1, IC50: 46 nM
LSD1, Ki: 30.3 nM
           
(1S,2R)-Tranylcypromine hydrochloride
KDM1/LSD1
           
LSD1-IN-22
KDM1/LSD1
           
LSD1-IN-39
LSD1, IC50: 0.18 μM
           
LSD1-IN-19
KDM1/LSD1
           
LSD1-IN-42
LSD1, IC50: 0.08 μM
           
LSD1/2-IN-3
KDM1/LSD1
           
Pulrodemstat hydrochloride
KDM1/LSD1
           
Tranylcypromine-d5 hydrochloride
KDM1/LSD1
           
AW4
LSD1
           
LSD1/HDAC-IN-1
LSD1, IC50: 0.571 μM
           
JQKD82        
KDM5
   
LSD1/ER-IN-1
KDM1/LSD1
           
LSD1-IN-36
LSD1, IC50: 0.8 nM
           
CBB1003 hydrochloride
KDM1/LSD1